Aminopterin (Why you need folic acid)

Special Saturday edition of MoTD: aminopterin.

i-d6061a4c87864ec299b61c34a2a6bdb7-aminopterin.gif

People have (quite understandably) been a little frantic about the putative taint found in pet food in recent days. Friday, ABC News reported that aminopterin was the contaminant, calling it "rat poison." I can't speak to the accuracy of the claim, but I can tell you that aminopterin isn't the kindest of molecules.

aminopterin, like the previously covered methotrexate, is a folate analogue that has found use in chemotherapy. Both work by impairing nucleic acid synthesis, and are quite toxic (the toxicity, unfortunately, shares the same origin as its efficacy in chemotherapy).

Tags

More like this

Apparently an FDA press conference this morning gave some bad news on pet food. See PetConnection.com The contamination may include dry food and other types of pet food than that originally reported. Initial reports were that only "savoury cuts" style wet food was at risk. Almost 10,000 deaths have…
Jonathan Wells recently gave a talk in Albuquerque at something called the "Forum on Science, Origins, and Design", a conference about which I can find absolutely nothing on the web. I wasn't there, of course, and I don't get invited to these goofy events anyway, but I did get a copy of Wells'…
Alternatively, "Despair of the Dork Side part 2". But I'd thought I'd stick with the Hamlet theme. So, no sooner does AW write not one but two barking mad posts about CO2 (see DotDS) than the what-I-had-thought-comparatively-sane Jo Nova complete the trilogy with It’s an Unsettling Climate for…
Janet Stemwedel is blogging, as is her wont, about questions of ethical behavior in science. She had a post Monday giving advice on how to counter unethical behavior, which all seems pretty good to me. Unfortunately, the people who read and comment on blogs about academic culture tend to start at "…

According to a very recent article, aminopterin is NOT used as a rat poison.
Someone patented its use as a rat poison in 1951, but it has never been used, it would degrade too fast --and be too costly to produce.

http://www.drugnewswire.com/14963/